GC34136
EPZ011989 trifluoroacetate
Also listed as EPZ011989 trifluoroacetate (EPZ-011989 trifluoroacetate)
EPZ-011989 trifluoroacetate is a potent and orally active Zeste Homolog 2 (EZH2) inhibitor with metabolic stability· EPZ-011989 trifluoroacetate has inhibitory inhibition for EZH2 with a Ki value of ＜3 nM· EPZ-011989 trifluoroacetate shows robust methyl mark inhibition and anti-tumor activity· EPZ-011989 trifluoroacetate can be used for the research of various cancers
ChemicalCAS1598383-41-5MW719.83FormulaC37H52F3N5O6
- CAS number
- 1598383-41-5
- Molecular weight
- 719.83
- Formula
- C37H52F3N5O6
- Solubility
- DMSO ： ≥ 34 mg/mL (47·23 mM)
- InChIKey
- JAUQBEFSKUVFDO-UHFFFAOYSA-N
- Catalogue number
- GC34136
- Brand
- GLPBIO
Computed properties PubChem CID 118704752 · TPSA 124 Ų · H-bond donors 3 · H-bond acceptors 12
- TPSA
- 124 Ų
- H-bond donors
- 3
- H-bond acceptors
- 12
- Rotatable bonds
- 12
- Heavy atoms
- 51
SMILES CCN(C1CCC(CC1)N(C)CCOC)C2=CC(=CC(=C2C)C(=O)NCC3=C(C=C(NC3=O)C)C)C#CCN4CCOCC4.C(=O)(C(F)(F)F)O
Computed descriptors from PubChem (CID 118704752), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il