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Chemical structure of EPZ-719

GC64343

EPZ-719

Also known as 4-fluoro-7-methyl-N-[(1R,3S)-3-[(3S)-3-[methyl(methylsulfonyl)amino]pyrrolidin-1-yl]cyclohexyl]-1H-indole-2-carboxamide

EPZ-719 is a novel and potent SETD2 inhibitor ( IC50 = 0·005 μM) with a high selectivity over other histone methyltransferases

ChemicalCAS2697176-16-0MW450.57FormulaC22H31FN4O3S
CAS number
2697176-16-0
Molecular weight
450.57
Formula
C22H31FN4O3S
InChIKey
ZLVKIBLQXFILMA-IKGGRYGDSA-N
Catalogue number
GC64343
Brand
GLPBIO
Computed properties PubChem CID 156599545 · XLogP 3 · TPSA 93.9 Ų · H-bond donors 2
XLogP
3
TPSA
93.9 Ų
H-bond donors
2
H-bond acceptors
6
Rotatable bonds
5
Heavy atoms
31

SMILES CC1=C2C(=C(C=C1)F)C=C(N2)C(=O)N[C@@H]3CCC[C@@H](C3)N4CC[C@@H](C4)N(C)S(=O)(=O)C

Computed descriptors from PubChem (CID 156599545), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.