
GC74088
EPZ011989 hydrochloride
Also known as N-[(4,6-dimethyl-2-oxo-1H-pyridin-3-yl)methyl]-3-[ethyl-[4-[2-methoxyethyl(methyl)amino]cyclohexyl]amino]-2-methyl-5-(3-morpholin-4-ylprop-1-ynyl)benzamide;hydrochloride
EPZ011989 drochloride is a potent and orally active Zeste Homolog 2 (EZH2) inhibitor, with a Ki value of <3 nM
ChemicalCAS2095432-26-9MW642.27FormulaC35H52ClN5O4
- CAS number
- 2095432-26-9
- Molecular weight
- 642.27
- Formula
- C35H52ClN5O4
- Solubility
- DMSO : 100 mg/mL (155·70 mM; Need ultrasonic)
- InChIKey
- LHRBDVKQGXCMQN-UHFFFAOYSA-N
- Catalogue number
- GC74088
- Brand
- GLPBIO
Computed properties PubChem CID 129896818 · TPSA 86.4 Ų · H-bond donors 3 · H-bond acceptors 7
- TPSA
- 86.4 Ų
- H-bond donors
- 3
- H-bond acceptors
- 7
- Rotatable bonds
- 12
- Heavy atoms
- 45
SMILES CCN(C1CCC(CC1)N(C)CCOC)C2=CC(=CC(=C2C)C(=O)NCC3=C(C=C(NC3=O)C)C)C#CCN4CCOCC4.Cl
Computed descriptors from PubChem (CID 129896818), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il