GC31614
GLPG0974
Also known as 4-[[(2R)-1-(1-benzothiophene-3-carbonyl)-2-methylazetidine-2-carbonyl]-[(3-chlorophenyl)methyl]amino]butanoic acid
GLPG0974 is an oral, high-affinity, potent and selective free fatty acid receptor 2 (FFA2, GPR43, IC50 = 9nM) antagonist
ChemicalCAS1391076-61-1MW485FormulaC25H25ClN2O4S
- CAS number
- 1391076-61-1
- Molecular weight
- 485
- Formula
- C25H25ClN2O4S
- Solubility
- DMSO ： 200 mg/mL (412·37 mM; Need ultrasonic)
- InChIKey
- MPMKMQHJHDHPBE-RUZDIDTESA-N
- Catalogue number
- GC31614
- Brand
- GLPBIO
Computed properties PubChem CID 57520598 · XLogP 4.3 · TPSA 106 Ų · H-bond donors 1
- XLogP
- 4.3
- TPSA
- 106 Ų
- H-bond donors
- 1
- H-bond acceptors
- 5
- Rotatable bonds
- 8
- Heavy atoms
- 33
SMILES C[C@@]1(CCN1C(=O)C2=CSC3=CC=CC=C32)C(=O)N(CCCC(=O)O)CC4=CC(=CC=C4)Cl
Computed descriptors from PubChem (CID 57520598), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il