GC65313
SSTR5 antagonist 1
Also known as 1-[2-[[3,5-diethoxy-4-(4-fluorophenyl)phenyl]methyl]-5-oxa-2,6-diazaspiro[3.4]oct-6-en-7-yl]piperidine-4-carboxylic acid
SSTR5 antagonist 1 is a potent, selective, and orally available somatostatin receptor subtype 5 (SSTR5) antagonist with IC50s of 9·6 and 57 nM for hSSTR5 and mSSTR5, respectively
ChemicalCAS1628741-91-2MW511.59FormulaC28H34FN3O5
- CAS number
- 1628741-91-2
- Molecular weight
- 511.59
- Formula
- C28H34FN3O5
- Solubility
- DMSO ： 90 mg/mL (175·92 mM; Need ultrasonic)
- InChIKey
- UQRAIIGEZLINAT-UHFFFAOYSA-N
- Catalogue number
- GC65313
- Brand
- GLPBIO
Computed properties PubChem CID 90423921 · XLogP 1.1 · TPSA 83.8 Ų · H-bond donors 1
- XLogP
- 1.1
- TPSA
- 83.8 Ų
- H-bond donors
- 1
- H-bond acceptors
- 8
- Rotatable bonds
- 9
- Heavy atoms
- 37
SMILES CCOC1=CC(=CC(=C1C2=CC=C(C=C2)F)OCC)CN3CC4(C3)CC(=NO4)N5CCC(CC5)C(=O)O
Computed descriptors from PubChem (CID 90423921), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il