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Chemical structure of EN1441

GC26841

EN1441

Also known as 6-chloro-3,3-dimethyl-4-prop-2-enoyl-1H-quinoxalin-2-one

EN1441 is a covalent degrader targeting the androgen receptor (AR) with an EC50 value of 4·2 μM and its truncated variant AR-V7

ChemicalCAS2196448-47-0MW264.71FormulaC13H13ClN2O2
CAS number
2196448-47-0
Molecular weight
264.71
Formula
C13H13ClN2O2
InChIKey
RSKGPRCITYZGEE-UHFFFAOYSA-N
Catalogue number
GC26841
Brand
GLPBIO
Computed properties PubChem CID 132317790 · XLogP 2.1 · TPSA 49.4 Ų · H-bond donors 1
XLogP
2.1
TPSA
49.4 Ų
H-bond donors
1
H-bond acceptors
2
Rotatable bonds
1
Heavy atoms
18

SMILES CC1(C(=O)NC2=C(N1C(=O)C=C)C=C(C=C2)Cl)C

Computed descriptors from PubChem (CID 132317790), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
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Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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