
GC15380
PF-562271
Also known as N-methyl-N-[3-[[[2-[(2-oxo-1,3-dihydroindol-5-yl)amino]-5-(trifluoromethyl)pyrimidin-4-yl]amino]methyl]-2-pyridinyl]methanesulfonamide
PF-562271 is a potent small-molecule inhibitor of focal adhesion kinase (FAK) and proline-rich tyrosine kinase 2 (Pyk2) with a IC50 of 1·5 and 14nmol/L, respectively
ChemicalCAS717907-75-0MW507.49FormulaC21H20F3N7O3S
- CAS number
- 717907-75-0
- Molecular weight
- 507.49
- Formula
- C21H20F3N7O3S
- Solubility
- ≥ 25·35mg/mL in DMSO, ≥ 2·25 mg/mL in EtOH with ultrasonic and warming
- InChIKey
- MZDKLVOWGIOKTN-UHFFFAOYSA-N
- Catalogue number
- GC15380
- Brand
- GLPBIO
Computed properties PubChem CID 11713159 · XLogP 2 · TPSA 138 Ų · H-bond donors 3
- XLogP
- 2
- TPSA
- 138 Ų
- H-bond donors
- 3
- H-bond acceptors
- 12
- Rotatable bonds
- 7
- Heavy atoms
- 35
SMILES CN(C1=C(C=CC=N1)CNC2=NC(=NC=C2C(F)(F)F)NC3=CC4=C(C=C3)NC(=O)C4)S(=O)(=O)C
Computed descriptors from PubChem (CID 11713159), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il