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Chemical structure of GB 83

GB40204

GB 83

Also known as N-[(2S)-3-cyclohexyl-1-[[(2S)-3-methyl-1-oxo-1-spiro[1,2-dihydroindene-3,4'-piperidine]-1'-ylpentan-2-yl]amino]-1-oxopropan-2-yl]-1,2-oxazole-5-carboxamide

Selective antagonist of human protease activated receptor 2 (PAR2) (IC50: 2 micromolar); reversibly inhibits PAR2 activation by both proteases and other PAR2 agonists

ChemicalCAS1252806-86-2MW548.72FormulaC32H44N4O4
CAS number
1252806-86-2
Molecular weight
548.72
Formula
C32H44N4O4
InChIKey
ZXMXAOYWSLZLQM-NZNGGYBSSA-N
Catalogue number
GB40204
Brand
GLPBIO
Computed properties PubChem CID 49843509 · XLogP 6.5 · TPSA 105 Ų · H-bond donors 2
XLogP
6.5
TPSA
105 Ų
H-bond donors
2
H-bond acceptors
5
Rotatable bonds
9
Heavy atoms
40

SMILES CCC(C)[C@@H](C(=O)N1CCC2(CCC3=CC=CC=C32)CC1)NC(=O)[C@H](CC4CCCCC4)NC(=O)C5=CC=NO5

Computed descriptors from PubChem (CID 49843509), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.