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Chemical structure of GSK973

GC92157

GSK973

Also known as (2S,3S)-2-(fluoromethyl)-7-N-methyl-5-N-[(1R,5S)-3-oxabicyclo[3.1.0]hexan-6-yl]-3-phenyl-2,3-dihydro-1-benzofuran-5,7-dicarboxamide

GSK620 is a bromodomain and extra terminal domain family of proteins (BET) bromodomain 2 (BD2) inhibitor (IC50s = 31·62, 15·85, 15·85, and 39·81 nM for BRD2, BRD3, BRD4, and BRDTBD2, respectively)

ChemicalCAS2138473-38-6MW410.4FormulaC23H23FN2O4
CAS number
2138473-38-6
Molecular weight
410.4
Formula
C23H23FN2O4
Solubility
Acetonitrile： Slightly soluble： 0·1–1 mg/ml,Methanol： Sparingly soluble： 1–10 mg/ml
InChIKey
WZQLVEPIBAOOGF-SFDMMAKQSA-N
Catalogue number
GC92157
Brand
GLPBIO
Computed properties PubChem CID 132004022 · XLogP 2.3 · TPSA 76.7 Ų · H-bond donors 2
XLogP
2.3
TPSA
76.7 Ų
H-bond donors
2
H-bond acceptors
5
Rotatable bonds
5
Heavy atoms
30

SMILES CNC(=O)C1=CC(=CC2=C1O[C@@H]([C@H]2C3=CC=CC=C3)CF)C(=O)NC4[C@H]5[C@@H]4COC5

Computed descriptors from PubChem (CID 132004022), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.