GC75712
PF-05214030
Also known as 4-[[1-(2,4-dichlorophenyl)sulfonyl-3-hydroxyazetidin-3-yl]methoxy]-2-fluorobenzonitrile
PF-05214030 is a TRPV4 antagonist (IC50: 4 and 27nM for hTRPV4 and rTRPV4 respectively)
ChemicalCAS1669444-50-1MW431.27FormulaC17H13Cl2FN2O4S
- CAS number
- 1669444-50-1
- Molecular weight
- 431.27
- Formula
- C17H13Cl2FN2O4S
- Solubility
- DMSO： 200 mg/mL (463·75 mM; Need ultrasonic)
- InChIKey
- RZAIRBXIVAVGHE-UHFFFAOYSA-N
- Catalogue number
- GC75712
- Brand
- GLPBIO
Computed properties PubChem CID 90665456 · XLogP 2.8 · TPSA 99 Ų · H-bond donors 1
- XLogP
- 2.8
- TPSA
- 99 Ų
- H-bond donors
- 1
- H-bond acceptors
- 7
- Rotatable bonds
- 5
- Heavy atoms
- 27
SMILES C1C(CN1S(=O)(=O)C2=C(C=C(C=C2)Cl)Cl)(COC3=CC(=C(C=C3)C#N)F)O
Computed descriptors from PubChem (CID 90665456), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il