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Chemical structure of NaV1·2/1·6 channel blocker-1

GC75469

NaV1·2/1·6 channel blocker-1

Also known as 2-methyl-3-propylimidazo[1,2-c][1,3]benzoxazine-5-thione

NaV1·2/1·6 channel blocker-1 is a potent NaV1·2/1·6 channel blocker, with IC50s of 9·8 and 24·4 μM for rNaV1·6 and hNaV1·2, respectively

ChemicalCAS1199944-04-1MW258.34FormulaC14H14N2OS
CAS number
1199944-04-1
Molecular weight
258.34
Formula
C14H14N2OS
Solubility
DMSO： 12·5 mg/mL (48·39 mM; ultrasonic and warming and heat to 60°C)
InChIKey
OEWGFBGGWFYYNM-UHFFFAOYSA-N
Catalogue number
GC75469
Brand
GLPBIO
Computed properties PubChem CID 101495288 · XLogP 3.8 · TPSA 59.1 Ų · H-bond donors 0
XLogP
3.8
TPSA
59.1 Ų
H-bond donors
0
H-bond acceptors
3
Rotatable bonds
2
Heavy atoms
18

SMILES CCCC1=C(N=C2N1C(=S)OC3=CC=CC=C32)C

Computed descriptors from PubChem (CID 101495288), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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