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Chemical structure of GSK360A

GC75037

GSK360A

Also known as 2-[[1-(2-cyclopropylethyl)-6-fluoro-4-hydroxy-2-oxoquinoline-3-carbonyl]amino]acetic acid

GSK360A is a potent and orally active HIF-PHD inhibitor with IC50 values of 10, 100, and 126 nM for PHD1, PHD2, and PHD3, respectively

ChemicalCAS931399-19-8MW348.33FormulaC17H17FN2O5
CAS number
931399-19-8
Molecular weight
348.33
Formula
C17H17FN2O5
Solubility
DMSO： 2 mg/mL (5·74 mM; Need ultrasonic and warming)
InChIKey
TYHRZQVUPPODPT-UHFFFAOYSA-N
Catalogue number
GC75037
Brand
GLPBIO
Computed properties PubChem CID 54685147 · XLogP 2.6 · TPSA 107 Ų · H-bond donors 3
XLogP
2.6
TPSA
107 Ų
H-bond donors
3
H-bond acceptors
6
Rotatable bonds
6
Heavy atoms
25

SMILES C1CC1CCN2C3=C(C=C(C=C3)F)C(=C(C2=O)C(=O)NCC(=O)O)O

Computed descriptors from PubChem (CID 54685147), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.