GC68803
BRD4 Inhibitor-20
Also known as 2-methoxy-N-(2-oxo-3-propan-2-ylidene-1H-indol-5-yl)benzenesulfonamide
BRD4 Inhibitor-20 is an effective inhibitor of the bromodomain-containing protein 4 (BRD4) with oral activity· It has inhibitory activity against both BRD4 (BD1) and BRD4 (BD2), with IC50 values of 19 nM and 28 nM, respectively· BRD4 Inhibitor-20 also exhibits anti-proliferative activity in cancer cell lines· It can be used for research on various cancers such as colon cancer
ChemicalCAS2490311-14-1MW358.41FormulaC18H18N2O4S
- CAS number
- 2490311-14-1
- Molecular weight
- 358.41
- Formula
- C18H18N2O4S
- Solubility
- DMSO ： 125 mg/mL (348·76 mM; ultrasonic and warming and heat to 60°C)
- InChIKey
- CDERLIUJSXSXFH-UHFFFAOYSA-N
- Catalogue number
- GC68803
- Brand
- GLPBIO
Computed properties PubChem CID 162653363 · XLogP 2.8 · TPSA 92.9 Ų · H-bond donors 2
- XLogP
- 2.8
- TPSA
- 92.9 Ų
- H-bond donors
- 2
- H-bond acceptors
- 5
- Rotatable bonds
- 4
- Heavy atoms
- 25
SMILES CC(=C1C2=C(C=CC(=C2)NS(=O)(=O)C3=CC=CC=C3OC)NC1=O)C
Computed descriptors from PubChem (CID 162653363), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il