Loading...
Chemical structure of PDK1-IN-RS2

GC66474

PDK1-IN-RS2

Also known as N-(6-chloro-1,3-benzothiazol-2-yl)-1-benzothiophene-2-sulfonamide

PDK1-IN-RS2 is a mimic of peptide docking motif (PIFtide) and is a substrate-selective PDK1 inhibitor with a Kd of 9 μM· PDK1-IN-RS2 suppresses the activation of the downstream kinases S6K1 by PDK1

ChemicalCAS1643958-89-7MW380.89FormulaC15H9ClN2O2S3
CAS number
1643958-89-7
Molecular weight
380.89
Formula
C15H9ClN2O2S3
Solubility
DMSO ： 125 mg/mL (328·18 mM; Need ultrasonic)
InChIKey
MZAVPBQCWWIYEQ-UHFFFAOYSA-N
Catalogue number
GC66474
Brand
GLPBIO
Computed properties PubChem CID 86290242 · XLogP 5.2 · TPSA 124 Ų · H-bond donors 1
XLogP
5.2
TPSA
124 Ų
H-bond donors
1
H-bond acceptors
6
Rotatable bonds
3
Heavy atoms
23

SMILES C1=CC=C2C(=C1)C=C(S2)S(=O)(=O)NC3=NC4=C(S3)C=C(C=C4)Cl

Computed descriptors from PubChem (CID 86290242), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.