Loading...
Chemical structure of CaV1·3 antagonist-1

GC65959

CaV1·3 antagonist-1

Also known as 1-[2-(3-chlorophenyl)ethyl]-3-cyclopentyl-1,3-diazinane-2,4,6-trione

CaV1·3 antagonist-1 is a potent and highly selective CaV1·3 L-type calcium channel (LTCC) antagonist with an IC50 of 1·7 μM· CaV1·3 antagonist-1 inhibits CaV1·3 LTCC >600-fold more potently than CaV1·2 LTCC· CaV1·3 antagonist-1, a cyclopentyl derivative, has the potential for Parkinson's disease research

ChemicalCAS1391385-57-1MW334.8FormulaC17H19ClN2O3
CAS number
1391385-57-1
Molecular weight
334.8
Formula
C17H19ClN2O3
Solubility
DMSO : 100 mg/mL (298·69 mM; Need ultrasonic)
InChIKey
AJKSBVCOTKODMF-UHFFFAOYSA-N
Catalogue number
GC65959
Brand
GLPBIO
Computed properties PubChem CID 57520395 · XLogP 3.1 · TPSA 57.7 Ų · H-bond donors 0
XLogP
3.1
TPSA
57.7 Ų
H-bond donors
0
H-bond acceptors
3
Rotatable bonds
4
Heavy atoms
23

SMILES C1CCC(C1)N2C(=O)CC(=O)N(C2=O)CCC3=CC(=CC=C3)Cl

Computed descriptors from PubChem (CID 57520395), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.