GC64999
MS402
Also known as 3-chloro-N-(4-methoxyphenyl)-4-[(2-methyl-3-oxocyclopenten-1-yl)amino]benzamide
MS402 is a BD1-selective BET BrD inhibitor with Kis of 77 nM, 718 nM, 110 nM, 200 nM, 83 nM, and 240 nM for BRD4(BD1), BRD4(BD2), BRD3(BD1), BRD3(BD2), BRD2(BD1) and BRD2(BD2), respectively
ChemicalCAS1672684-68-2MW370.83FormulaC20H19ClN2O3
- CAS number
- 1672684-68-2
- Molecular weight
- 370.83
- Formula
- C20H19ClN2O3
- Solubility
- DMSO ： 100 mg/mL (269·67 mM; Need ultrasonic)
- InChIKey
- VZTVTSICPINUNG-UHFFFAOYSA-N
- Catalogue number
- GC64999
- Brand
- GLPBIO
Computed properties PubChem CID 90718189 · XLogP 3.6 · TPSA 67.4 Ų · H-bond donors 2
- XLogP
- 3.6
- TPSA
- 67.4 Ų
- H-bond donors
- 2
- H-bond acceptors
- 4
- Rotatable bonds
- 5
- Heavy atoms
- 26
SMILES CC1=C(CCC1=O)NC2=C(C=C(C=C2)C(=O)NC3=CC=C(C=C3)OC)Cl
Computed descriptors from PubChem (CID 90718189), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il