GC62630
TAS-117 hydrochloride
TAS-117 hydrochloride is a potent, selective, orally active allosteric Akt inhibitor (with IC50s of 4·8, 1·6, and 44 nM for Akt1, 2, and 3, respectively)· TAS-117 hydrochloride triggers anti-myeloma activities and enhances fatal endoplasmic reticulum (ER) stress induced by proteasome inhibition· TAS-117 hydrochloride induces apoptosis and autophagy
ChemicalMW460.96FormulaC26H25ClN4O2
- CAS number
- —
- Molecular weight
- 460.96
- Formula
- C26H25ClN4O2
- Solubility
- DMSO ： 62·5 mg/mL (135·59 mM; ultrasonic and warming and heat to 60°C)
- Catalogue number
- GC62630
- Brand
- GLPBIO
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il