
GC36652
MPT0B392
Also known as 6-methoxy-2-(3,4,5-trimethoxyphenyl)sulfonylquinolin-5-amine
MPT0B392, an orally active quinoline derivative, induces c-Jun N-terminal kinase (JNK) activation, leading to apoptosis· MPT0B392 inhibits tubulin polymerization and triggers induction of the mitotic arrest, followed by mitochondrial membrane potential loss and caspases cleavage by activation of JNK and ultimately leads to apoptosis· MPT0B392 is demonstrated to be a novel microtubule-depolymerizing agent and enhances the cytotoxicity of sirolimus in sirolimus-resistant acute leukemic cells and the multidrug resistant cell line
- CAS number
- 1346169-92-3
- Molecular weight
- 404.44
- Formula
- C19H20N2O6S
- Solubility
- Soluble in DMSO
- InChIKey
- RBBRZMLZQCYQJM-UHFFFAOYSA-N
- Catalogue number
- GC36652
- Brand
- GLPBIO
Computed properties PubChem CID 56834893 · XLogP 2.5 · TPSA 118 Ų · H-bond donors 1
- XLogP
- 2.5
- TPSA
- 118 Ų
- H-bond donors
- 1
- H-bond acceptors
- 8
- Rotatable bonds
- 6
- Heavy atoms
- 28
SMILES COC1=C(C2=C(C=C1)N=C(C=C2)S(=O)(=O)C3=CC(=C(C(=C3)OC)OC)OC)N
Computed descriptors from PubChem (CID 56834893), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il