GC36142
GK921
Also known as 3-(2-phenylethynyl)-2-(2-pyrrolidin-1-ylethoxy)pyrido[2,3-b]pyrazine
GK921 is a transglutaminase 2 (TGase) inhibitor with an IC50 of 7·71 μM for human recombinant TGase 2
ChemicalCAS1025015-40-0MW344.41FormulaC21H20N4O
- CAS number
- 1025015-40-0
- Molecular weight
- 344.41
- Formula
- C21H20N4O
- Solubility
- DMSO： ≥ 30 mg/mL (87·11 mM)
- InChIKey
- MNYJJHBAEYKXEG-UHFFFAOYSA-N
- Catalogue number
- GC36142
- Brand
- GLPBIO
Computed properties PubChem CID 56682080 · XLogP 3.4 · TPSA 51.1 Ų · H-bond donors 0
- XLogP
- 3.4
- TPSA
- 51.1 Ų
- H-bond donors
- 0
- H-bond acceptors
- 5
- Rotatable bonds
- 6
- Heavy atoms
- 26
SMILES C1CCN(C1)CCOC2=NC3=C(N=CC=C3)N=C2C#CC4=CC=CC=C4
Computed descriptors from PubChem (CID 56682080), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il