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Chemical structure of ERK5-IN-2

GC36002

ERK5-IN-2

Also known as 4-(2-bromo-6-fluorobenzoyl)-N-pyridin-3-yl-1H-pyrrole-2-carboxamide

ERK5-IN-2 is an orally active, sub-micromolar, selective ERK5 inhibitor with IC50s of 0·82 μM, 3 μM for ERK5 and ERK5 MEF2D, respectively

ChemicalCAS1888305-96-1MW388.19FormulaC17H11BrFN3O2
CAS number
1888305-96-1
Molecular weight
388.19
Formula
C17H11BrFN3O2
Solubility
DMSO： 250 mg/mL (644·01 mM)
InChIKey
ATKCERYALDNMPL-UHFFFAOYSA-N
Catalogue number
GC36002
Brand
GLPBIO
Computed properties PubChem CID 118959080 · XLogP 2.9 · TPSA 74.9 Ų · H-bond donors 2
XLogP
2.9
TPSA
74.9 Ų
H-bond donors
2
H-bond acceptors
4
Rotatable bonds
4
Heavy atoms
24

SMILES C1=CC(=C(C(=C1)Br)C(=O)C2=CNC(=C2)C(=O)NC3=CN=CC=C3)F

Computed descriptors from PubChem (CID 118959080), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.