Loading...
Chemical structure of Protein kinase inhibitors 1

GC34131

Protein kinase inhibitors 1

Also known as (5E)-5-[[6-oxo-5-(6-piperazin-1-yl-3-pyridinyl)-1H-pyridin-3-yl]methylidene]-1,3-thiazolidine-2,4-dione

Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9·5 nM

ChemicalCAS1365986-44-2MW383.42FormulaC18H17N5O3S
CAS number
1365986-44-2
Molecular weight
383.42
Formula
C18H17N5O3S
Solubility
Soluble in DMSO
InChIKey
YHUKWWWCNSTFHL-RIYZIHGNSA-N
Catalogue number
GC34131
Brand
GLPBIO
Computed properties PubChem CID 132274054 · XLogP 0.4 · TPSA 129 Ų · H-bond donors 3
XLogP
0.4
TPSA
129 Ų
H-bond donors
3
H-bond acceptors
7
Rotatable bonds
3
Heavy atoms
27

SMILES C1CN(CCN1)C2=NC=C(C=C2)C3=CC(=CNC3=O)/C=C/4\C(=O)NC(=O)S4

Computed descriptors from PubChem (CID 132274054), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.