GC31505
MCHr1 antagonist 2
Also known as N-[1-(1,3-benzodioxol-5-ylmethyl)piperidin-4-yl]-6-fluoro-4-oxochromene-2-carboxamide
MCHR1 antagonist 2 is an antagonist of melanin concentrating hormone receptor 1, with an IC50 of 65 nM; MCHR1 antagonist 2 also inhibits hERG, with an IC50 of 4·0 nM in IMR-32 cells
ChemicalCAS863115-70-2MW424.42FormulaC23H21FN2O5
- CAS number
- 863115-70-2
- Molecular weight
- 424.42
- Formula
- C23H21FN2O5
- Solubility
- DMSO ： 10 mg/mL (23·56 mM; ultrasonic and adjust pH to 6 with HCl)
- InChIKey
- HHCYCBKPWYJVEB-UHFFFAOYSA-N
- Catalogue number
- GC31505
- Brand
- GLPBIO
Computed properties PubChem CID 11464405 · XLogP 3 · TPSA 77.1 Ų · H-bond donors 1
- XLogP
- 3
- TPSA
- 77.1 Ų
- H-bond donors
- 1
- H-bond acceptors
- 7
- Rotatable bonds
- 4
- Heavy atoms
- 31
SMILES C1CN(CCC1NC(=O)C2=CC(=O)C3=C(O2)C=CC(=C3)F)CC4=CC5=C(C=C4)OCO5
Computed descriptors from PubChem (CID 11464405), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il