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Chemical structure of GSK4028

GC30714

GSK4028

Also known as 4-bromo-2-methyl-5-[[(3S,5S)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-one

GSK4028 is the enantiomeric negative control of GSK4027, which is a PCAF/GCN5 bromodomain chemical probe, the pIC50 of GSK4028 is 4·9 in a time-resolved fluorescence resonance energy transfer (TR-FRET) assay

ChemicalCAS2079886-19-2MW377.28FormulaC17H21BrN4O
CAS number
2079886-19-2
Molecular weight
377.28
Formula
C17H21BrN4O
Solubility
DMSO ： 100 mg/mL (265·06 mM; Need ultrasonic)
InChIKey
VZAFGXCWAWRULT-KGLIPLIRSA-N
Catalogue number
GC30714
Brand
GLPBIO
Computed properties PubChem CID 132941768 · XLogP 2.5 · TPSA 47.9 Ų · H-bond donors 1
XLogP
2.5
TPSA
47.9 Ų
H-bond donors
1
H-bond acceptors
4
Rotatable bonds
3
Heavy atoms
23

SMILES CN1C[C@@H](C[C@@H](C1)NC2=C(C(=O)N(N=C2)C)Br)C3=CC=CC=C3

Computed descriptors from PubChem (CID 132941768), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.