Loading...
Chemical structure of GSK 2193874

GC16917

GSK 2193874

Also known as 7-bromo-N-(1-phenylcyclopropyl)-3-[(4-piperidin-1-ylpiperidin-1-yl)methyl]-2-[3-(trifluoromethyl)phenyl]quinoline-4-carboxamide

TRPV4 antagonist, potent and selective

ChemicalCAS1336960-13-4MW691.62FormulaC37H38BrF3N4O
CAS number
1336960-13-4
Molecular weight
691.62
Formula
C37H38BrF3N4O
Solubility
DMF： 15 mg/mL,DMSO： 14 mg/mL,Ethanol： 15 mg/mL,Ethanol：PBS (pH 7·2)(1：2)： 0·3 mg/mL
InChIKey
UIVOZBSCHXCGPS-UHFFFAOYSA-N
Catalogue number
GC16917
Brand
GLPBIO
Computed properties PubChem CID 53464483 · XLogP 7.8 · TPSA 48.5 Ų · H-bond donors 1
XLogP
7.8
TPSA
48.5 Ų
H-bond donors
1
H-bond acceptors
7
Rotatable bonds
7
Heavy atoms
46

SMILES C1CCN(CC1)C2CCN(CC2)CC3=C(C4=C(C=C(C=C4)Br)N=C3C5=CC(=CC=C5)C(F)(F)F)C(=O)NC6(CC6)C7=CC=CC=C7

Computed descriptors from PubChem (CID 53464483), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.