
GA21358
DABCYL-TNF-α-EDANS (-4 to +6) (human)
Also known as 5-[2-[[2-[[2-[[2-[[2-[[2-[[2-[2-[[5-amino-2-[2-[[2-[[4-[[4-(dimethylamino)phenyl]diazenyl]benzoyl]amino]-4-methylpentanoyl]amino]propanoylamino]-5-oxopentanoyl]amino]propanoylamino]-3-methylbutanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxypropanoyl]amino]-3-hydroxypropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]ethylamino]naphthalene-1-sulfonic acid
The FRET substrate DABCYL-LAQAVRSSSR-EDANS represents the optimal size for efficient fluorescent quenching, while incorporating all of the necessary amino acids to yield a viable substrate to be used for rapid screening of compounds for inhibition of TNF-α converting enzyme (TACE, ADAM17 endopeptidase) activity
- CAS number
- 396716-14-6
- Molecular weight
- 1573.8
- Formula
- C70H104N22O18S
- Solubility
- Soluble in DMSO
- InChIKey
- NLLNLPZJUJVHNC-UHFFFAOYSA-N
- Catalogue number
- GA21358
- Brand
- GLPBIO
Computed properties PubChem CID 165365314 · XLogP -2.2 · TPSA 655 Ų · H-bond donors 21
- XLogP
- -2.2
- TPSA
- 655 Ų
- H-bond donors
- 21
- H-bond acceptors
- 24
- Rotatable bonds
- 46
- Heavy atoms
- 111
SMILES CC(C)CC(C(=O)NC(C)C(=O)NC(CCC(=O)N)C(=O)NC(C)C(=O)NC(C(C)C)C(=O)NC(CCCN=C(N)N)C(=O)NC(CO)C(=O)NC(CO)C(=O)NC(CO)C(=O)NC(CCCN=C(N)N)C(=O)NCCNC1=CC=CC2=C1C=CC=C2S(=O)(=O)O)NC(=O)C3=CC=C(C=C3)N=NC4=CC=C(C=C4)N(C)C
Computed descriptors from PubChem (CID 165365314), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il