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Chemical structure of Kv2·1-IN-1

GC75728

Kv2·1-IN-1

Also known as 2-ethoxy-N-[1-[3-(methylamino)phenyl]ethyl]-5-(2-methylpropanoylamino)benzamide

Kv2·1-IN-1 (compound 80) is a potent inhibitor of Kv2·1, with the IC50 value of 0·07 μM, selectivity >130 fold over other K+, Na+, and Ca2+ ion channels

ChemicalCAS2252448-93-2MW383.48FormulaC22H29N3O3
CAS number
2252448-93-2
Molecular weight
383.48
Formula
C22H29N3O3
Solubility
DMSO： 100 mg/mL (260·77 mM; Need ultrasonic)
InChIKey
SVTYEIYBHHWMJJ-UHFFFAOYSA-N
Catalogue number
GC75728
Brand
GLPBIO
Computed properties PubChem CID 141731038 · XLogP 3.6 · TPSA 79.5 Ų · H-bond donors 3
XLogP
3.6
TPSA
79.5 Ų
H-bond donors
3
H-bond acceptors
4
Rotatable bonds
8
Heavy atoms
28

SMILES CCOC1=C(C=C(C=C1)NC(=O)C(C)C)C(=O)NC(C)C2=CC(=CC=C2)NC

Computed descriptors from PubChem (CID 141731038), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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