Loading...
Chemical structure of Enerisant

GC74093

Enerisant

Also known as [1-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]pyrazol-4-yl]-morpholin-4-ylmethanone

Enerisant is a potent, selective, competitive and orally active histamine H3 receptor antagonist/inverse agonist with IC50s of 2·89 nM and 14·5 nM against human and rat histamine H3 receptors

ChemicalCAS1152747-82-4MW398.5FormulaC22H30N4O3
CAS number
1152747-82-4
Molecular weight
398.5
Formula
C22H30N4O3
Solubility
DMSO ： 100 mg/mL (250·94 mM; Need ultrasonic)
InChIKey
IABXVJILZYNSTM-GOSISDBHSA-N
Catalogue number
GC74093
Brand
GLPBIO
Computed properties PubChem CID 42601503 · XLogP 2.3 · TPSA 59.8 Ų · H-bond donors 0
XLogP
2.3
TPSA
59.8 Ų
H-bond donors
0
H-bond acceptors
5
Rotatable bonds
7
Heavy atoms
29

SMILES C[C@@H]1CCCN1CCCOC2=CC=C(C=C2)N3C=C(C=N3)C(=O)N4CCOCC4

Computed descriptors from PubChem (CID 42601503), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.