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Chemical structure of Enerisant hydrochloride

GC71523

Enerisant hydrochloride

Also known as [1-[4-[3-[(2R)-2-methylpyrrolidin-1-yl]propoxy]phenyl]pyrazol-4-yl]-morpholin-4-ylmethanone;hydrochloride

Enerisant (TS-091) hydrochloride is a potent, highly selective, competitive and orally active histamine H3 receptor antagonist/inverse agonist with IC50s of 2·89 nM and 14·5 nM against human and rat histamine H3 receptors, respectively

ChemicalCAS1152749-07-9MW434.96FormulaC22H31ClN4O3
CAS number
1152749-07-9
Molecular weight
434.96
Formula
C22H31ClN4O3
Solubility
DMSO ： 50 mg/mL (114·95 mM; ultrasonic and warming and heat to 60°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
InChIKey
QVMTVPSORZKQPZ-GMUIIQOCSA-N
Catalogue number
GC71523
Brand
GLPBIO
Computed properties PubChem CID 66933564 · TPSA 59.8 Ų · H-bond donors 1 · H-bond acceptors 5
TPSA
59.8 Ų
H-bond donors
1
H-bond acceptors
5
Rotatable bonds
7
Heavy atoms
30

SMILES C[C@@H]1CCCN1CCCOC2=CC=C(C=C2)N3C=C(C=N3)C(=O)N4CCOCC4.Cl

Computed descriptors from PubChem (CID 66933564), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.