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Chemical structure of STAT3-SH2 domain inhibitor 1

GC73355

STAT3-SH2 domain inhibitor 1

Also known as [4-[(4-cyclohexylphenyl)methyl-[2-[methyl-(2,3,4,5,6-pentafluorophenyl)sulfonylamino]acetyl]amino]phenyl]boronic acid

STAT3-SH2 domain inhibitor 1 is a potent Src Homology 2 (SH2) Domain of STAT3 (STAT3-SH2 domain) inhibitor with a Kd value of 1·57 μM

ChemicalCAS2816059-41-1MW610.4FormulaC28H28BF5N2O5S
CAS number
2816059-41-1
Molecular weight
610.4
Formula
C28H28BF5N2O5S
Solubility
DMSO ： 8·33 mg/mL (13·65 mM; ultrasonic and warming and heat to 80°C)
InChIKey
CEZFPVMURCGETD-UHFFFAOYSA-N
Catalogue number
GC73355
Brand
GLPBIO
Computed properties PubChem CID 165413024 · TPSA 107 Ų · H-bond donors 2 · H-bond acceptors 11
TPSA
107 Ų
H-bond donors
2
H-bond acceptors
11
Rotatable bonds
9
Heavy atoms
42

SMILES B(C1=CC=C(C=C1)N(CC2=CC=C(C=C2)C3CCCCC3)C(=O)CN(C)S(=O)(=O)C4=C(C(=C(C(=C4F)F)F)F)F)(O)O

Computed descriptors from PubChem (CID 165413024), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.