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Chemical structure of ZEN-2759

GC72992

ZEN-2759

Also known as 1-benzyl-5-(3,5-dimethyl-1,2-oxazol-4-yl)pyridin-2-one

ZEN-2759 is a potent BET (Bromodomain and Extra-Terminal Domain) inhibitor, with IC50 values of 0·23, 0·08 and 0·28 μM for BRD4(BD1), BRD4(BD2), and BRD4(BD1BD2), respectively

ChemicalCAS1616400-50-0MW280.32FormulaC17H16N2O2
CAS number
1616400-50-0
Molecular weight
280.32
Formula
C17H16N2O2
Solubility
DMSO ： 100 mg/mL (356·74 mM; Need ultrasonic)
InChIKey
CIJOVPIWGFQZFF-UHFFFAOYSA-N
Catalogue number
GC72992
Brand
GLPBIO
Computed properties PubChem CID 76683643 · XLogP 2.3 · TPSA 46.3 Ų · H-bond donors 0
XLogP
2.3
TPSA
46.3 Ų
H-bond donors
0
H-bond acceptors
3
Rotatable bonds
3
Heavy atoms
21

SMILES CC1=C(C(=NO1)C)C2=CN(C(=O)C=C2)CC3=CC=CC=C3

Computed descriptors from PubChem (CID 76683643), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.