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Chemical structure of TRPV2-selective blocker 1

GC71419

TRPV2-selective blocker 1

Also known as 5-(1,3-dithiolan-2-ylidene)-4-methyl-5-phenylpentan-2-one

TRPV2-selective blocker 1 (compound IV2-1) is a selective TRPV2 channel blocker with an IC50 of 6·3 μM

ChemicalCAS2242724-49-6MW278.43FormulaC15H18OS2
CAS number
2242724-49-6
Molecular weight
278.43
Formula
C15H18OS2
Solubility
DMSO : 100 mg/mL (359·16 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
InChIKey
RCALJRZMLQRHLX-UHFFFAOYSA-N
Catalogue number
GC71419
Brand
GLPBIO
Computed properties PubChem CID 133053728 · XLogP 3.9 · TPSA 67.7 Ų · H-bond donors 0
XLogP
3.9
TPSA
67.7 Ų
H-bond donors
0
H-bond acceptors
3
Rotatable bonds
4
Heavy atoms
18

SMILES CC(CC(=O)C)C(=C1SCCS1)C2=CC=CC=C2

Computed descriptors from PubChem (CID 133053728), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.