GC71181
Glucocorticoid receptor modulator 1
Also known as N-(1-benzoyl-3,4-dihydro-2H-quinolin-6-yl)-5-chloro-2-methoxy-4-methylbenzenesulfonamide
Glucocorticoid receptor modulator 1 is a highly potent and orally active non-steroidal selective glucocorticoid receptor modulator with an IC50 value of 9 nM and 130 nM for NF-κB and AP-1, respectively
ChemicalCAS2868357-11-1MW470.97FormulaC24H23ClN2O4S
- CAS number
- 2868357-11-1
- Molecular weight
- 470.97
- Formula
- C24H23ClN2O4S
- Solubility
- DMSO ： 100 mg/mL (212·33 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
- InChIKey
- BDARZHMPJRWQLB-UHFFFAOYSA-N
- Catalogue number
- GC71181
- Brand
- GLPBIO
Computed properties PubChem CID 166176961 · XLogP 4.8 · TPSA 84.1 Ų · H-bond donors 1
- XLogP
- 4.8
- TPSA
- 84.1 Ų
- H-bond donors
- 1
- H-bond acceptors
- 5
- Rotatable bonds
- 5
- Heavy atoms
- 32
SMILES CC1=CC(=C(C=C1Cl)S(=O)(=O)NC2=CC3=C(C=C2)N(CCC3)C(=O)C4=CC=CC=C4)OC
Computed descriptors from PubChem (CID 166176961), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il