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Chemical structure of BMS 182874

GC70458

BMS 182874

Also known as 5-(dimethylamino)-N-(3,4-dimethyl-1,2-oxazol-5-yl)naphthalene-1-sulfonamide

BMS 182874 is an orallyactive, highly selective endothelin receptor (ETA receptor) antagonist, with IC50 value of 0·150 μM, Ki of 0·055 μM

ChemicalCAS153042-42-3MW345.42FormulaC17H19N3O3S
CAS number
153042-42-3
Molecular weight
345.42
Formula
C17H19N3O3S
Solubility
DMSO ： 125 mg/mL (361·88 mM; Need ultrasonic; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
InChIKey
MJRGSRRZKSJHOE-UHFFFAOYSA-N
Catalogue number
GC70458
Brand
GLPBIO
Computed properties PubChem CID 122272 · XLogP 3.4 · TPSA 83.8 Ų · H-bond donors 1
XLogP
3.4
TPSA
83.8 Ų
H-bond donors
1
H-bond acceptors
6
Rotatable bonds
4
Heavy atoms
24

SMILES CC1=C(ON=C1C)NS(=O)(=O)C2=CC=CC3=C2C=CC=C3N(C)C

Computed descriptors from PubChem (CID 122272), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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