
GC65178
KB-5492 free base
Also known as (4-methoxyphenyl) 2-[4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-1-yl]acetate
KB-5492 free base is a potent and selective inhibitor of sigma receptor, inhibits specific [3H]1,3-di(2-tolyl)guanidine (DTG) binding to the sigma receptor with an IC50 of 3·15 μM
ChemicalCAS113594-64-2MW430.49FormulaC23H30N2O6
- CAS number
- 113594-64-2
- Molecular weight
- 430.49
- Formula
- C23H30N2O6
- Solubility
- DMSO : 100 mg/mL (232·29 mM; Need ultrasonic)
- InChIKey
- RVYZAZTXLLAVGZ-UHFFFAOYSA-N
- Catalogue number
- GC65178
- Brand
- GLPBIO
Computed properties PubChem CID 131083 · XLogP 2.9 · TPSA 69.7 Ų · H-bond donors 0
- XLogP
- 2.9
- TPSA
- 69.7 Ų
- H-bond donors
- 0
- H-bond acceptors
- 8
- Rotatable bonds
- 10
- Heavy atoms
- 31
SMILES COC1=CC=C(C=C1)OC(=O)CN2CCN(CC2)CC3=CC(=C(C(=C3)OC)OC)OC
Computed descriptors from PubChem (CID 131083), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il