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Chemical structure of GSK5182

GC64453

GSK5182

Also known as 4-[(Z)-1-[4-[2-(dimethylamino)ethoxy]phenyl]-5-hydroxy-2-phenylpent-1-enyl]phenol

GSK5182 is a highly selective and orally active inverse agonist of estrogen-related receptor γ (ERRγ) with an IC50 of 79 nM

ChemicalCAS877387-37-6MW417.54FormulaC27H31NO3
CAS number
877387-37-6
Molecular weight
417.54
Formula
C27H31NO3
Solubility
DMSO ： 25 mg/mL (59·87 mM; ultrasonic and warming and heat to 80°C)
InChIKey
ZVSFNBNLNLXEFQ-RQZHXJHFSA-N
Catalogue number
GC64453
Brand
GLPBIO
Computed properties PubChem CID 6852176 · XLogP 5.9 · TPSA 52.9 Ų · H-bond donors 2
XLogP
5.9
TPSA
52.9 Ų
H-bond donors
2
H-bond acceptors
4
Rotatable bonds
10
Heavy atoms
31

SMILES CN(C)CCOC1=CC=C(C=C1)/C(=C(/CCCO)\C2=CC=CC=C2)/C3=CC=C(C=C3)O

Computed descriptors from PubChem (CID 6852176), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.