GC62555
Setd2-IN-1 tfa
Also listed as EZM0414 (SETD2-IN-1) TFA
EZM0414 (SETD2-IN-1) TFA is the TFA salt (Trifluoroacetate) form of EZM0414· EZM0414 is a first-in-class, potent, selective, orally bioavailable small molecule inhibitor of the enzymatic activity of SETD2 with an IC50 value of 18nM
ChemicalCAS2411759-92-5MW514.51FormulaC24H30F4N4O4
- CAS number
- 2411759-92-5
- Molecular weight
- 514.51
- Formula
- C24H30F4N4O4
- Solubility
- DMSO ： 200 mg/mL (388·72 mM; Need ultrasonic)
- InChIKey
- HASNOYOGMISGTP-PPPUBMIESA-N
- Catalogue number
- GC62555
- Brand
- GLPBIO
Computed properties PubChem CID 155971202 · TPSA 106 Ų · H-bond donors 3 · H-bond acceptors 9
- TPSA
- 106 Ų
- H-bond donors
- 3
- H-bond acceptors
- 9
- Rotatable bonds
- 3
- Heavy atoms
- 36
SMILES CC1=C2C(=C(C=C1)F)C=C(N2)C(=O)N[C@@H]3CCC[C@@H](C3)N4CCN(CC4)C(=O)C.C(=O)(C(F)(F)F)O
Computed descriptors from PubChem (CID 155971202), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il