GC62276
CP-609754
Also known as 6-[(R)-(4-chlorophenyl)-hydroxy-(3-methylimidazol-4-yl)methyl]-4-(3-ethynylphenyl)-1-methylquinolin-2-one
CP-609754 (LNK-754) is a potent and reversible farnesyltransferase inhibitor with potential anticancer activity·The IC50 for inhibiting farnesylation of recombinant human H-Ras is 0·57 ng/mL and recombinant K-Ras is 46 ng/mL
ChemicalCAS1190094-64-4MW479.96FormulaC29H22ClN3O2
- CAS number
- 1190094-64-4
- Molecular weight
- 479.96
- Formula
- C29H22ClN3O2
- Solubility
- DMSO ： 100 mg/mL (208·35 mM; Need ultrasonic)
- InChIKey
- JAHDAIPFBPPQHQ-GDLZYMKVSA-N
- Catalogue number
- GC62276
- Brand
- GLPBIO
Computed properties PubChem CID 46208720 · XLogP 4 · TPSA 58.4 Ų · H-bond donors 1
- XLogP
- 4
- TPSA
- 58.4 Ų
- H-bond donors
- 1
- H-bond acceptors
- 3
- Rotatable bonds
- 5
- Heavy atoms
- 35
SMILES CN1C=NC=C1[C@@](C2=CC=C(C=C2)Cl)(C3=CC4=C(C=C3)N(C(=O)C=C4C5=CC=CC(=C5)C#C)C)O
Computed descriptors from PubChem (CID 46208720), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il