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Chemical structure of ER 819762

GC50722

ER 819762

Also known as (5S)-1'-[(3,5-dimethylphenyl)methyl]-2-ethyl-6,8-dimethoxy-5-methylspiro[5,10-dihydroimidazo[1,5-b][2]benzazepine-3,4'-piperidine]-1-one

ER 819762 is an orally active, highly selective prostaglandin E2 (PGE2) EP4 receptor antagonist with an EC50 of 70 nM against human EP4 receptor

ChemicalCAS1155773-15-1MW489.65FormulaC30H39N3O3
CAS number
1155773-15-1
Molecular weight
489.65
Formula
C30H39N3O3
Solubility
ethanol|2·45|5withgentlewarming|DMSO|0·98|2withgentlewarming|
InChIKey
ANKFBAJRCGOKJJ-QFIPXVFZSA-N
Catalogue number
GC50722
Brand
GLPBIO
Computed properties PubChem CID 42596951 · XLogP 4.5 · TPSA 45.3 Ų · H-bond donors 0
XLogP
4.5
TPSA
45.3 Ų
H-bond donors
0
H-bond acceptors
4
Rotatable bonds
5
Heavy atoms
36

SMILES CCN1C(=O)N2CC3=C([C@H](C=C2C14CCN(CC4)CC5=CC(=CC(=C5)C)C)C)C(=CC(=C3)OC)OC

Computed descriptors from PubChem (CID 42596951), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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