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Chemical structure of SB-242084 (hydrochloride)

GC44875

SB-242084 (hydrochloride)

Also known as 6-chloro-5-methyl-N-[6-[(2-methyl-3-pyridinyl)oxy]-3-pyridinyl]-2,3-dihydroindole-1-carboxamide;dihydrochloride

SB 242084 hydrochloride is a 5-HT2C receptor antagonist(pKi=9·0) that displays 158- and 100-fold selectivity over 5-HT2A and 5-HT2B receptors respectively

ChemicalCAS1049747-87-6MW467.8FormulaC21H19ClN4O2•2HCl
CAS number
1049747-87-6
Molecular weight
467.8
Formula
C21H19ClN4O2•2HCl
Solubility
DMF： 30 mg/ml,DMSO： 30 mg/ml,Ethanol： 1 mg/ml,PBS (pH 7·2)： 10 mg/ml
InChIKey
GCMNSEILNIPNSX-UHFFFAOYSA-N
Catalogue number
GC44875
Brand
GLPBIO
Computed properties PubChem CID 16219981 · TPSA 67.4 Ų · H-bond donors 3 · H-bond acceptors 4
TPSA
67.4 Ų
H-bond donors
3
H-bond acceptors
4
Rotatable bonds
3
Heavy atoms
30

SMILES CC1=CC2=C(C=C1Cl)N(CC2)C(=O)NC3=CN=C(C=C3)OC4=C(N=CC=C4)C.Cl.Cl

Computed descriptors from PubChem (CID 16219981), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.