GC42955
BMS 986122
Also known as 2-(3-bromo-4-methoxyphenyl)-3-(4-chlorophenyl)sulfonyl-1,3-thiazolidine
BMS 986122 is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1 human osteosarcoma cells expressing μ-opioid receptors (EC50 = 3 μM)
ChemicalCAS313669-88-4MW448.8FormulaC16H15BrClNO3S2
- CAS number
- 313669-88-4
- Molecular weight
- 448.8
- Formula
- C16H15BrClNO3S2
- Solubility
- DMF： 10 mg/ml,DMSO： 10 mg/ml,DMSO：PBS (pH 7·2) (1：1)： 0·5 mg/ml,Ethanol： 2 mg/ml
- InChIKey
- PNGJPVDGZNPZHY-UHFFFAOYSA-N
- Catalogue number
- GC42955
- Brand
- GLPBIO
Computed properties PubChem CID 4644453 · XLogP 4.4 · TPSA 80.3 Ų · H-bond donors 0
- XLogP
- 4.4
- TPSA
- 80.3 Ų
- H-bond donors
- 0
- H-bond acceptors
- 5
- Rotatable bonds
- 4
- Heavy atoms
- 24
SMILES COC1=C(C=C(C=C1)C2N(CCS2)S(=O)(=O)C3=CC=C(C=C3)Cl)Br
Computed descriptors from PubChem (CID 4644453), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il