
GC37725
TAK-960 dihydrochloride
TAK-960 dihydrochloride is an orally available, selective inhibitor of polo-like kinase 1 (PLK1), with an IC50 of 0·8 nM· TAK-960 dihydrochloride also shows inhibitory activities against PLK2 and PLK3, with IC50s of 16·9 and 50·2 nM, respectively· TAK-960 dihydrochloride inhibits proliferation of multiple cancer cell lines and exhibits significant efficacy against multiple tumor xenografts
ChemicalMW634.52FormulaC27H36Cl2F3N7O3
- CAS number
- —
- Molecular weight
- 634.52
- Formula
- C27H36Cl2F3N7O3
- Solubility
- DMSO: ≥ 98·57 mg/mL (155·35 mM)
- Catalogue number
- GC37725
- Brand
- GLPBIO
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il