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Chemical structure of FAPI-4

GC36029

FAPI-4

Also known as 2-[4,7-bis(carboxymethyl)-10-[2-[4-[3-[4-[[2-[(2S)-2-cyano-4,4-difluoropyrrolidin-1-yl]-2-oxoethyl]carbamoyl]quinolin-6-yl]oxypropyl]piperazin-1-yl]-2-oxoethyl]-1,4,7,10-tetrazacyclododec-1-yl]acetic acid

FAPI-4 is a potent fibroblast activation protein (FAP) inhibitor for the targeting FAP· FAPI-4 can be used in cancer research· 68Ga-FAPI-4 PET/CT is a promising new diagnostic method for imaging various kinds of cancer, with good tumor-to-background contrast ratios

ChemicalCAS2374782-02-0MW872.91FormulaC40H54F2N10O10
CAS number
2374782-02-0
Molecular weight
872.91
Formula
C40H54F2N10O10
Solubility
DMSO： 100 mg/mL (114·56 mM)
InChIKey
ICWDAESAANBIGG-LJAQVGFWSA-N
Catalogue number
GC36029
Brand
GLPBIO
Computed properties PubChem CID 138454803 · XLogP -6.8 · TPSA 244 Ų · H-bond donors 4
XLogP
-6.8
TPSA
244 Ų
H-bond donors
4
H-bond acceptors
19
Rotatable bonds
16
Heavy atoms
62

SMILES C1CN(CCN1CCCOC2=CC3=C(C=CN=C3C=C2)C(=O)NCC(=O)N4CC(C[C@H]4C#N)(F)F)C(=O)CN5CCN(CCN(CCN(CC5)CC(=O)O)CC(=O)O)CC(=O)O

Computed descriptors from PubChem (CID 138454803), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.