GC17473
Pelitinib
Also listed as Pelitinib (EKB-569)
Pelitinib (EKB-569) (EKB-569;WAY-EKB 569) is an irreversible inhibitor of EGFR with an IC50 of 38·5 nM; also slightly inhibits Src, MEK/ERK and ErbB2 with IC50s of 282, 800, and 1255 nM, respectively
ChemicalCAS257933-82-7MW467.92FormulaC24H23ClFN5O2
- CAS number
- 257933-82-7
- Molecular weight
- 467.92
- Formula
- C24H23ClFN5O2
- Solubility
- ≥ 11·7mg/mL in DMSO
- InChIKey
- WVUNYSQLFKLYNI-AATRIKPKSA-N
- Catalogue number
- GC17473
- Brand
- GLPBIO
Computed properties PubChem CID 6445562 · XLogP 4.5 · TPSA 90.3 Ų · H-bond donors 2
- XLogP
- 4.5
- TPSA
- 90.3 Ų
- H-bond donors
- 2
- H-bond acceptors
- 7
- Rotatable bonds
- 8
- Heavy atoms
- 33
SMILES CCOC1=C(C=C2C(=C1)N=CC(=C2NC3=CC(=C(C=C3)F)Cl)C#N)NC(=O)/C=C/CN(C)C
Computed descriptors from PubChem (CID 6445562), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il