
GC10463
SB 216763
Also known as 3-(2,4-dichlorophenyl)-4-(1-methylindol-3-yl)pyrrole-2,5-dione
SB 216763 stands out as a powerful, selective, and ATP-competitive inhibitor of GSK-3, effectively targeting both GSK-3α and GSK-3β with an impressive IC50 of 34·3 nM[1-3]
ChemicalCAS280744-09-4MW371.22FormulaC19H12Cl2N2O2
- CAS number
- 280744-09-4
- Molecular weight
- 371.22
- Formula
- C19H12Cl2N2O2
- Solubility
- ≥ 56·8mg/mL in DMSO
- InChIKey
- JCSGFHVFHSKIJH-UHFFFAOYSA-N
- Catalogue number
- GC10463
- Brand
- GLPBIO
Computed properties PubChem CID 176158 · XLogP 3.9 · TPSA 51.1 Ų · H-bond donors 1
- XLogP
- 3.9
- TPSA
- 51.1 Ų
- H-bond donors
- 1
- H-bond acceptors
- 2
- Rotatable bonds
- 2
- Heavy atoms
- 25
SMILES CN1C=C(C2=CC=CC=C21)C3=C(C(=O)NC3=O)C4=C(C=C(C=C4)Cl)Cl
Computed descriptors from PubChem (CID 176158), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il