
GB40161
CS1
Also known as 4-(6-hydroxynaphthalen-2-yl)benzene-1,2-diol
TOPO IIα inhibitor with broad-spectrum in vitro antitumor effects (IC50 values 4·3 µM, 11·5 µM, and 4·6 µM for inhibition of proliferation of breast cancer MDA-MB-231, human lung cancer A549 and human cervical cancer HeLa cell lines, respectively)· CS1 functions as a Topo II poison to stabilize Topo II/DNA complex, which leads to DNA damage, cell cycle arrest at G2/M phase and apoptosis, and is 6-10-fold less cytotoxic against HL7702 and HUVEC cells compared with etoposide
- CAS number
- 1448009-94-6
- Molecular weight
- 252.26
- Formula
- C16H12O3
- InChIKey
- LDFFDYWHCCDSBO-UHFFFAOYSA-N
- Catalogue number
- GB40161
- Brand
- GLPBIO
Computed properties PubChem CID 57173257 · XLogP 3.7 · TPSA 60.7 Ų · H-bond donors 3
- XLogP
- 3.7
- TPSA
- 60.7 Ų
- H-bond donors
- 3
- H-bond acceptors
- 3
- Rotatable bonds
- 1
- Heavy atoms
- 19
SMILES C1=CC2=C(C=CC(=C2)O)C=C1C3=CC(=C(C=C3)O)O
Computed descriptors from PubChem (CID 57173257), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il