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Chemical structure of BQ-610

GA21190

BQ-610

Also known as (2R)-2-[[(2R)-2-[[(2S)-2-(azepane-1-carbonylamino)-4-methylpentanoyl]amino]-3-(1-formylindol-3-yl)propanoyl]amino]-3-(1H-indol-3-yl)propanoic acid

BQ-610 is a very potent ET-A receptor antagonist which is about 30000 times more selective for ET-A receptors than for ET-B receptors· Furthermore, it has been found that BQ-610 strongly antagonizes ET-1 induced concentration in porcine coronary artery with a pA? value of 8·2

ChemicalCAS141595-53-1MW656.78FormulaC36H44N6O6
CAS number
141595-53-1
Molecular weight
656.78
Formula
C36H44N6O6
Solubility
Soluble in DMSO
InChIKey
QHSRPPJQBFQWSC-OJDZSJEKSA-N
Catalogue number
GA21190
Brand
GLPBIO
Computed properties PubChem CID 123905 · XLogP 4.8 · TPSA 166 Ų · H-bond donors 5
XLogP
4.8
TPSA
166 Ų
H-bond donors
5
H-bond acceptors
6
Rotatable bonds
12
Heavy atoms
48

SMILES CC(C)C[C@@H](C(=O)N[C@H](CC1=CN(C2=CC=CC=C21)C=O)C(=O)N[C@H](CC3=CNC4=CC=CC=C43)C(=O)O)NC(=O)N5CCCCCC5

Computed descriptors from PubChem (CID 123905), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
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