GC75858
Lumateperone
Also known as 1-(4-fluorophenyl)-4-[(10R,15S)-4-methyl-1,4,12-triazatetracyclo[7.6.1.05,16.010,15]hexadeca-5,7,9(16)-trien-12-yl]butan-1-one
Lumateperone (ITI-007) is an orally active 5-HT2A receptor antagonist (Ki = 0·54 nM), a partial agonist of presynaptic D2 receptors and an antagonist of postsynaptic D2 receptors (Ki = 32 nM), and a dopamine D1 receptor modulator
ChemicalCAS313368-91-1MW393.5FormulaC24H28FN3O
- CAS number
- 313368-91-1
- Molecular weight
- 393.5
- Formula
- C24H28FN3O
- Solubility
- DMSO： 125 mg/mL (317·66 mM; Need ultrasonic)
- InChIKey
- HOIIHACBCFLJET-SFTDATJTSA-N
- Catalogue number
- GC75858
- Brand
- GLPBIO
Computed properties PubChem CID 21302490 · XLogP 3.8 · TPSA 26.8 Ų · H-bond donors 0
- XLogP
- 3.8
- TPSA
- 26.8 Ų
- H-bond donors
- 0
- H-bond acceptors
- 5
- Rotatable bonds
- 5
- Heavy atoms
- 29
SMILES CN1CCN2[C@H]3CCN(C[C@H]3C4=C2C1=CC=C4)CCCC(=O)C5=CC=C(C=C5)F
Computed descriptors from PubChem (CID 21302490), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.
Ordering in Israel
- Lead time
- Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
- Pricing
- Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
- Documents
- Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
- Who we serve
- Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.
- Questions
- WhatsApp · +972-55-990-7576 · orders@labo.co.il