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Chemical structure of GRK2 Inhibitor 2

GC75632

GRK2 Inhibitor 2

Also known as 2-[(3-methoxyphenyl)methyl]-7-(1H-pyrazol-4-yl)phthalazin-1-one

GRK2 Inhibitor 2 is an orally active and selective G protein-coupled receptor kinase 2 (GRK) inhibitor with an IC50 of 19 nM

ChemicalCAS2592436-21-8MW332.36FormulaC19H16N4O2
CAS number
2592436-21-8
Molecular weight
332.36
Formula
C19H16N4O2
Solubility
DMSO： 100 mg/mL (300·88 mM; Need ultrasonic)
InChIKey
CYINSAOYPJZRPS-UHFFFAOYSA-N
Catalogue number
GC75632
Brand
GLPBIO
Computed properties PubChem CID 155594167 · XLogP 2.3 · TPSA 70.6 Ų · H-bond donors 1
XLogP
2.3
TPSA
70.6 Ų
H-bond donors
1
H-bond acceptors
4
Rotatable bonds
4
Heavy atoms
25

SMILES COC1=CC=CC(=C1)CN2C(=O)C3=C(C=CC(=C3)C4=CNN=C4)C=N2

Computed descriptors from PubChem (CID 155594167), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
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Pricing
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Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
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