Loading...
Chemical structure of FR194921

GC72870

FR194921

Also known as 2-(1-methylpiperidin-4-yl)-6-(2-phenylpyrazolo[1,5-a]pyridin-3-yl)pyridazin-3-one

FR194921 is a potent, selective and orally active and cross the blood-brain barrier Adenosine A1 antagonist with Ki value of 6·6, 5400 nM for A1, A2A, respectively

ChemicalCAS202646-80-8MW385.46FormulaC23H23N5O
CAS number
202646-80-8
Molecular weight
385.46
Formula
C23H23N5O
Solubility
DMSO ： 2 mg/mL (5·19 mM; Need ultrasonic and warming)
InChIKey
YHDRUTMZCJZJAL-UHFFFAOYSA-N
Catalogue number
GC72870
Brand
GLPBIO
Computed properties PubChem CID 9821511 · XLogP 2.8 · TPSA 53.2 Ų · H-bond donors 0
XLogP
2.8
TPSA
53.2 Ų
H-bond donors
0
H-bond acceptors
4
Rotatable bonds
3
Heavy atoms
29

SMILES CN1CCC(CC1)N2C(=O)C=CC(=N2)C3=C4C=CC=CN4N=C3C5=CC=CC=C5

Computed descriptors from PubChem (CID 9821511), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.