Loading...
Chemical structure of CB1/2 agonist 1

GC71002

CB1/2 agonist 1

Also known as 5-bromo-N-cycloheptyl-1-[(4-fluorophenyl)methyl]-6-methyl-2-oxopyridine-3-carboxamide

CB1/2 agonist 1 is a potent and cross the blood-brain barrier CB1/2 agonist with EC50s of 56·15, 11·63 nM for CB1R and CB2R, respectively

ChemicalCAS2986688-90-6MW435.33FormulaC21H24BrFN2O2
CAS number
2986688-90-6
Molecular weight
435.33
Formula
C21H24BrFN2O2
Solubility
DMSO ： 20 mg/mL (45·94 mM; ultrasonic and warming and heat to 70°C; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
InChIKey
IBDOGMBSQPMZKN-UHFFFAOYSA-N
Catalogue number
GC71002
Brand
GLPBIO
Computed properties PubChem CID 162654853 · XLogP 4.6 · TPSA 49.4 Ų · H-bond donors 1
XLogP
4.6
TPSA
49.4 Ų
H-bond donors
1
H-bond acceptors
3
Rotatable bonds
4
Heavy atoms
27

SMILES CC1=C(C=C(C(=O)N1CC2=CC=C(C=C2)F)C(=O)NC3CCCCCC3)Br

Computed descriptors from PubChem (CID 162654853), public domain. Identity cross-checked against the supplier's molecular formula and weight — verify before use.

Ordering in Israel

Lead time
Ships from the manufacturer to your lab in 8–14 business days; customs and cold chain handled by LABO Scientific.
Pricing
Quoted in ILS, excl. VAT. Add the item to your quote and we confirm the final price, usually the same business day.
Documents
Lot certificate of analysis and manufacturer SDS are emailed with your order confirmation.
Who we serve
Universities, hospitals and biotech companies across Israel. Research use only — not for diagnostic or therapeutic use.